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重新利用药物靶向端粒酶:发现雷替曲塞(Raltitrexed)的抗癌潜力
为解决端粒酶(Telomerase)靶向治疗难题,研究人员开展药物重利用研究,发现雷替曲塞有抑制潜力。 端粒酶(Telomerase)是一种与癌症的复制永生有关的逆转录酶,由于其结构复杂且缺乏临床批准的小分子抑制剂,它一直是治疗干预的难题。在这项研究中 ...
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